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Amphetamine is known to inhibit monoamine oxidase, whereas the flexibility of amphetamine and its metabolites to inhibit several P450 isozymes along with other enzymes hasn't been adequately elucidated. In vitro experiments with human microsomes suggest slight inhibition of CYP2D6 by amphetamine and insignificant inhibition of CYP1A2, 2D6, and 3A4